An expedient synthesis of substituted indoles
作者： Amos B. Smith , Melean Visnick
DOI: 10.1016/S0040-4039(00)89243-6
关键词:
摘要: Abstract Condensation of carboxylic acid esters with organodilithium reagents derived from N-trimethylsilyl-o-toluidine or N-trimethylsilyl-o-ethyl aniline affords substituted indoles.
elsevier.com
sci-hub.se 参考文章(13)
A.H. Jackson, P. Smith, Electrophilic substitution in indoles—III: Rearrangement of 3,3-dialkyl indolenines Tetrahedron. ,vol. 24, pp. 2227- 2239 ,(1968) , 10.1016/0040-4020(68)88125-6
Paul A. Wender, Alan W. White, Methodology for indole synthesis Tetrahedron Letters. ,vol. 22, pp. 1475- 1478 ,(1981) , 10.1016/S0040-4039(01)90354-5
Wayland E. Noland, Kent R. Rush, Lowell R. Smith, Nitration of Indoles. IV. The Nitration of 2-Phenylindole1 Journal of Organic Chemistry. ,vol. 31, pp. 65- 69 ,(1966) , 10.1021/JO01339A013
Robert E. Ludt, Gary P. Crowther, Charles R. Hauser, Effect of tetramethylethylenediamine on the metalation of o- and p-N,N-dimethyltoluidines with n-butyllithium. Deuteration and electrophilic condensation of intermediate lithioamines The Journal of Organic Chemistry. ,vol. 35, pp. 1288- 1296 ,(1970) , 10.1021/JO00830A009
Masao Nakazaki, Twofold Wagner-Meerwein Type Rearrangement of 2,3-Disubstituted Indoles Bulletin of the Chemical Society of Japan. ,vol. 33, pp. 461- 465 ,(1960) , 10.1246/BCSJ.33.461
Hugo Illy, Lance Funderburk, Fischer indole synthesis. Direction of cyclization of isopropylmethyl ketone phenylhydrazone Journal of Organic Chemistry. ,vol. 33, pp. 4283- 4285 ,(1968) , 10.1021/JO01275A066
Paul G. Gassman, William N. Schenk, The use of [2,3] sigmatropic rearrangements for the specific ortho-substitution of polycyclic aromatic amines. The methylation of naphthylamines and the synthesis of 1H-benz[g]indoles and 3H-benz[e]indoles Journal of Organic Chemistry. ,vol. 42, pp. 3240- 3243 ,(1977) , 10.1021/JO00440A008
A.Ian Scott, Biogenetic-type synthesis of the indole alkaloids Bioorganic Chemistry. ,vol. 3, pp. 398- 429 ,(1974) , 10.1016/0045-2068(74)90011-X
R. J. P. CORRIU, J. J. E. MOREAU, Some Uses of Silicon-Nitrogen Bonds in Organic Synthesis ChemInform. ,vol. 16, ,(1985) , 10.1002/CHIN.198506376
Yoshihiko Ito, Kazuhiro Kobayashi, Norihiko Seko, Takeo Saegusa, Indole syntheses utilizing o-methylphenyl isocyanides. Bulletin of the Chemical Society of Japan. ,vol. 57, pp. 73- 84 ,(1984) , 10.1246/BCSJ.57.73