Process for producing fingolimod salts

作者: Ramesh Matioram Gidwani , Channaveerayya Hiremath

DOI:

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摘要: The invention relates to a process for producing pharmaceutically acceptable salts of fingolimod (I), comprising the step reacting N-[1,1-bis hydroxymethyl-3-(4-octyl phenyl)-propyl]-acylamide (II) with an acidic compound. Furthermore, provides different and polymorphic form hydrochloride.

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