Synthesis and Antitubercular, Antimicrobial, and Hemolytic Activity of Methyl D-Glucopyranuronate and Its Simplest Derivatives
作者： M. G. Belenok , O. V. Andreeva , B. F. Garifullin , A. S. Strobykina , M. A. Kravchenko
DOI: 10.1134/S1070363217120106
关键词:
摘要: Methyl glucuronate and some of its simplest derivatives have been synthesized, their antitubercular, antimicrobial, hemolytic activities studied. The glucuronic acid shown for the first time to exhibit a high antitubercular activity which is comparable with isoniazid.
springer.com
sci-hub.se 参考文章(47)
LA Baltina, RM Kondratenko, SR Mustafina, OB Flekhter, Yu I Murinov, VA Davydova, FS Zarudii, AF Ismagilova, GA Tolstikov, None, Synthesis of Glycyrrhizic Acid from Glycyrram and Pharmaciological Characterization of the Product Pharmaceutical Chemistry Journal. ,vol. 35, pp. 40- 44 ,(2001) , 10.1023/A:1010454810888
Zygmunt Sidorczyk, Anna N. Kondakova, Krystyna Zych, Sof'ya N. Senchenkova, Alexander S. Shashkov, Dominika Drzewiecka, Yuriy A. Knirel, Structure of the O-polysaccharide from Proteus myxofaciens: Classification of the bacterium into a new Proteus O-serogroup FEBS Journal. ,vol. 270, pp. 3182- 3188 ,(2003) , 10.1046/J.1432-1033.2003.03698.X
Stanislav G. Batrakov, Denis I. Nikitin, Irina A. Pitryuk, A novel glycolipid, 1,2-diacyl-3-alpha-D-glucuronopyranosyl-sn-glycerol taurineamide, from the budding seawater bacterium Hyphomonas jannaschiana. Biochimica et Biophysica Acta. ,vol. 1302, pp. 167- 176 ,(1996) , 10.1016/0005-2760(96)00060-4
Matthew A Wikler, None, Methods for dilution antimicrobial susceptibility tests for bacteria that grow aerobically : Approved standard CLSI (NCCLS). ,vol. 26, ,(2006)
Wayne Pilgrim, Paul V. Murphy, SnCl4- and TiCl4-Catalyzed Anomerization of Acylated O- and S-Glycosides: Analysis of Factors That Lead to Higher α:β Anomer Ratios and Reaction Rates Journal of Organic Chemistry. ,vol. 75, pp. 6747- 6755 ,(2010) , 10.1021/JO101090F
Ta-Chun Cheng, Steve R. Roffler, Shey-Cherng Tzou, Kuo-Hsiang Chuang, Yu-Cheng Su, Chih-Hung Chuang, Chien-Han Kao, Chien-Shu Chen, I-Hong Harn, Kuan-Yi Liu, Tian-Lu Cheng, Yu-Ling Leu, An Activity-Based Near-Infrared Glucuronide Trapping Probe for Imaging β-Glucuronidase Expression in Deep Tissues Journal of the American Chemical Society. ,vol. 134, pp. 3103- 3110 ,(2012) , 10.1021/JA209335Z
Fátima Paiva-Martins, Aníbal Silva, Vasco Almeida, Mafalda Carvalheira, Cristina Serra, José Enrique Rodrígues-Borges, João Fernandes, Luis Belo, Alice Santos-Silva, Protective activity of hydroxytyrosol metabolites on erythrocyte oxidative-induced hemolysis. Journal of Agricultural and Food Chemistry. ,vol. 61, pp. 6636- 6642 ,(2013) , 10.1021/JF4016202
Jean-Claude Florent, Xia Dong, Gilbert Gaudel, Sofia Mitaku, Claude Monneret, Jean-Pierre Gesson, Jean-Claude Jacquesy, Martine Mondon, Brigitte Renoux, Solo Andrianomenjanahary, Sylvie Michel, Michel Koch, François Tillequin, Manfred Gerken, Joerg Czech, Rainer Straub, Klaus Bosslet, Prodrugs of Anthracyclines for Use in Antibody-Directed Enzyme Prodrug Therapy Journal of Medicinal Chemistry. ,vol. 41, pp. 3572- 3581 ,(1998) , 10.1021/JM970589L
Ahmed I. Khodair, Philippe Bertrand, A new approach to the synthesis of substituted 4-imidazolidinones as potential antiviral and antitumor agents Tetrahedron. ,vol. 54, pp. 4859- 4872 ,(1998) , 10.1016/S0040-4020(98)00170-7
Yuqiang Wang, Huiling Yuan, Susan C Wright, Hong Wang, James W Larrick, Synthesis and preliminary cytotoxicity study of glucuronide derivatives of CC-1065 analogues Bioorganic & Medicinal Chemistry. ,vol. 11, pp. 1569- 1575 ,(2003) , 10.1016/S0968-0896(02)00603-X