Irreversible enzyme inhibitors. 101. A modified synthesis of 2-substituted-4,6-diamino-1,2-dihydro-2-methyl-1-phenyl-s-triazines†
作者： B. R. Baker , Morris A. Johnson
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sci-hub.se 参考文章(15)
B.R. Baker, Factors in the Design of Active-Site-Directed Irreversible Inhibitors Journal of Pharmaceutical Sciences. ,vol. 53, pp. 347- 364 ,(1964) , 10.1002/JPS.2600530402
F. H. S. Curd, F. L. Rose, 71. Synthetic antimalarials. Part IV. 2-Phenylguanidino-4-aminoalkylamino-6-methylpyrimidines Journal of the Chemical Society (Resumed). pp. 362- 366 ,(1946) , 10.1039/JR9460000362
B.R. Baker, Beng-Thong Ho, Differential Inhibition of Dihydrofolic Reductase from Different Species Journal of Pharmaceutical Sciences. ,vol. 53, pp. 1137- 1138 ,(1964) , 10.1002/JPS.2600530943
B.R. Baker, Howard S. Shapiro, Irreversible Enzyme Inhibitors LXXI Journal of Pharmaceutical Sciences. ,vol. 56, pp. 33- 38 ,(1967) , 10.1002/JPS.2600560106
B. R. Baker, Beng-Thong Ho, Thomas Neilson, Analogs of tetrahydrofolic acid. XII. On the relative contribution by the 2-amino and 4-hydroxy groups of 2-amino-5-(3-anilinopropyl)-6-methyl-4-pyrimidinol to inhibition of folic reductase and thymidylate synthetase Journal of Heterocyclic Chemistry. ,vol. 1, pp. 79- 87 ,(1964) , 10.1002/JHET.5570010206
B.R. Baker, Rich B. Meyer, Irreversible Enzyme Inhibitors LXXXIV Journal of Pharmaceutical Sciences. ,vol. 56, pp. 570- 576 ,(1967) , 10.1002/JPS.2600560505
B.R. Baker, Beng-Thong Ho, Daniel V. Santi, Analogs of Tetrahydrofolic Acid XXVII Journal of Pharmaceutical Sciences. ,vol. 54, pp. 1415- 1424 ,(1965) , 10.1002/JPS.2600541005
B. R. Baker, Johannes H. Jordaan, Irreversible enzyme inhibitors. LXXXIII. Candidate active-site-directed irreversible inhibitors of dihydrofolic reductase. VIII. Derivatives of 2,4-diaminopyrimidine. II†‡ Journal of Heterocyclic Chemistry. ,vol. 4, pp. 31- 38 ,(1967) , 10.1002/JHET.5570040106
B.R. Baker, William W. Lee, Ethel Tong, Non-classical antimetabolites. VI. 4-(Iodoacetamido)-salicylic acid, an exo-alkylating irreversible inhibitor Journal of Theoretical Biology. ,vol. 3, pp. 459- 483 ,(1962) , 10.1016/S0022-5193(62)80037-X
B. R. Baker, Beng-Thong Ho, Analogs of tetrahydrofolic acid. XXIII. 1-(ω-phenylalkyl)-4,6-diamino-1,2-dihydro-s-triazines as inhibitors of dihydrofolic reductase†‡ Journal of Heterocyclic Chemistry. ,vol. 2, pp. 72- 79 ,(1965) , 10.1002/JHET.5570020113