Intramolecular cyclization of S-alkyl derivatives of aminomercaptoimidazoles and -benzimidazoles as a method for the annulation of the thiadiazine ring
作者： N. I. Gaponenko , A. A. Kolodina , A. V. Lesin , S. V. Kurbatov
DOI: 10.1007/S11172-012-0157-8
关键词:
摘要: A method was developed for the annulation of tetrahydrothiadiazine moiety to imidazole and benzimidazole rings through intramolecular cyclization S-alkyl derivatives aminomercaptoimidazoles -benzimidazoles. The factors controlling stereoselectivity formation ring were revealed.
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