Activation of α-sp3 centres toward electrophilic substitution in alcohols and amines

作者: Alan R. Katritzky , Saumitra Sengupta

DOI: 10.1007/BF02839447

关键词:

摘要: The scope of electrophilic substitution at alpha-sp3 centres in alcohols and amines via their alpha-lithio species is reviewed. importance alpha-activation by the hetero atom protecting group deliniated with special reference to transient protection-activation methodology.

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