1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study
作者： Mubarak H Shaikh , Dnyaneshwar D Subhedar , Laxman Nawale , Dhiman Sarkar , Firoz A Kalam Khan
DOI: 10.1039/C5MD00057B
关键词:
摘要: A library of thirty one 1,2,3-triazole derivatives efficiently preparedviaclick chemistry and evaluated for their antitubercular, antioxidant, and cytotoxic activities.
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sci-hub.se 参考文章(52)
Yuan H. Zhao, Michael H. Abraham, Joelle Le, Anne Hersey, Chris N. Luscombe, Gordon Beck, Brad Sherborne, Ian Cooper, Rate-limited steps of human oral absorption and QSAR studies. Pharmaceutical Research. ,vol. 19, pp. 1446- 1457 ,(2002) , 10.1023/A:1020444330011
Albert Padwa, 1,3-Dipolar Cycloaddition Chemistry ,(1984)
Fauzia Mir, Syed Shafi, MS Zaman, Nitin Pal Kalia, Vikrant S Rajput, Chaitanya Mulakayala, Naveen Mulakayala, Inshad A Khan, MS Alam, None, Sulfur rich 2-mercaptobenzothiazole and 1,2,3-triazole conjugates as novel antitubercular agents European Journal of Medicinal Chemistry. ,vol. 76, pp. 274- 283 ,(2014) , 10.1016/J.EJMECH.2014.02.017
Christian W. Tornøe, Caspar Christensen, Morten Meldal, Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(i)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides. Journal of Organic Chemistry. ,vol. 67, pp. 3057- 3064 ,(2002) , 10.1021/JO011148J
Jean Paul Dzoyem, Santosh Kumar Guru, Constant Anatole Pieme, Victor Kuete, Akash Sharma, Inshad Ali Khan, Ajit Kumar Saxena, Ram Anuj Vishwakarma, None, Cytotoxic and antimicrobial activity of selected Cameroonian edible plants. BMC Complementary and Alternative Medicine. ,vol. 13, pp. 78- 78 ,(2013) , 10.1186/1472-6882-13-78
Upasana Singh, Shamim Akhtar, Abhishek Mishra, Dhiman Sarkar, A novel screening method based on menadione mediated rapid reduction of tetrazolium salt for testing of anti-mycobacterial agents Journal of Microbiological Methods. ,vol. 84, pp. 202- 207 ,(2011) , 10.1016/J.MIMET.2010.11.013
Kurt V. Gothelf, Karl Anker Jørgensen, Asymmetric 1,3-Dipolar Cycloaddition Reactions Chemical Reviews. ,vol. 98, pp. 863- 910 ,(1998) , 10.1021/CR970324E
Jaiprakash N Sangshetti, Rehan I Shaikh, Firoz A Kalam Khan, Rajendra H Patil, Sayali D Marathe, Wasudev N Gade, Devanand B Shinde, None, Synthesis, antileishmanial activity and docking study of N'-substitutedbenzylidene-2-(6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)acetohydrazides. Bioorganic & Medicinal Chemistry Letters. ,vol. 24, pp. 1605- 1610 ,(2014) , 10.1016/J.BMCL.2014.01.035
G. Ciapetti, E. Cenni, L. Pratelli, A. Pizzoferrato, In vitro evaluation of cell/biomaterial interaction by MTT assay. Biomaterials. ,vol. 14, pp. 359- 364 ,(1993) , 10.1016/0142-9612(93)90055-7
Sandip G. Agalave, Suleman R. Maujan, Vandana S. Pore, Click Chemistry: 1,2,3‐Triazoles as Pharmacophores Chemistry-an Asian Journal. ,vol. 6, pp. 2696- 2718 ,(2011) , 10.1002/ASIA.201100432