‘Click’ synthesis of cobalt bis(dicarbollide)–cholesterol conjugates

作者: Anna A. Druzina , Akim V. Shmalko , Ekaterina P. Andreichuk , Olga B. Zhidkova , Irina D. Kosenko

DOI: 10.1016/J.MENCOM.2019.11.007

关键词:

摘要: New conjugates of cholesterol and cobalt bis(dicarbollide) were synthesized using ‘click’ cycloaddition 3b-(2-azidoethyl) cholest-5-ene acetylene-equipped bis(dicarbollides). The boronated cholesterols can be interest for liposomal drug delivery boron neutron capture therapy cancer.

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