Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate Receptors
作者： Craig W. Lindsley , Kyle A. Emmitte , Corey R. Hopkins , Thomas M. Bridges , Karen J. Gregory
DOI: 10.1021/ACS.CHEMREV.5B00656
关键词:
摘要: … Allosteric modulation of GPCRs has initiated a new era of … Allosteric ligands stabilize unique conformations of the GPCR … of the basics of GPCR allosteric pharmacology, medicinal …
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