3,5-T2 Is an Alternative Ligand for the Thyroid Hormone Receptor β1
作者： A. Mendoza , P. Navarrete-Ramírez , G. Hernández-Puga , P. Villalobos , G. Holzer
DOI: 10.1210/EN.2013-1030
关键词:
摘要: … with 17β-estradiol for binding to ERβ in the prostate, the growth of … and 3βAdiol for VDR and ERβ, respectively, an alternative … Schematic representation of the putative action mechanism …
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endojournals.org参考文章(43)
Pan Wang, Yujing Wen, Gui-Zhen Han, Pritam Kaur Sidhu, Bao Ting Zhu, Characterization of the oestrogenic activity of non-aromatic steroids: are there male-specific endogenous oestrogen receptor modulators? British Journal of Pharmacology. ,vol. 158, pp. 1796- 1807 ,(2009) , 10.1111/J.1476-5381.2009.00467.X
C Horst, H Rokos, H J Seitz, Rapid stimulation of hepatic oxygen consumption by 3,5-di-iodo-L-thyronine. Biochemical Journal. ,vol. 261, pp. 945- 950 ,(1989) , 10.1042/BJ2610945
M A Lazar, T J Berrodin, H P Harding, Differential DNA binding by monomeric, homodimeric, and potentially heteromeric forms of the thyroid hormone receptor. Molecular and Cellular Biology. ,vol. 11, pp. 5005- 5015 ,(1991) , 10.1128/MCB.11.10.5005
A. Lanni, M. Moreno, A. Lombardi, F. Goglia, Rapid stimulation in vitro of rat liver cytochrome oxidase activity by 3,5-diiodo-L-thyronine and by 3,3'-diiodo-L-thyronine Molecular and Cellular Endocrinology. ,vol. 99, pp. 89- 94 ,(1994) , 10.1016/0303-7207(94)90150-3
SG Ball, J Sokolov, WW Chin, 3,5-Diiodo-L-thyronine (T2) has selective thyromimetic effects in vivo and in vitro Journal of Molecular Endocrinology. ,vol. 19, pp. 137- 147 ,(1997) , 10.1677/JME.0.0190137
Anthony N. Hollenberg, Tsuyoshi Monden, Fredric E. Wondisford, Ligand-independent and -dependent Functions of Thyroid Hormone Receptor Isoforms Depend upon Their Distinct Amino Termini Journal of Biological Chemistry. ,vol. 270, pp. 14274- 14280 ,(1995) , 10.1074/JBC.270.24.14274
Hinrich Gronemeyer, Jan-Åke Gustafsson, Vincent Laudet, Principles for modulation of the nuclear receptor superfamily Nature Reviews Drug Discovery. ,vol. 3, pp. 950- 964 ,(2004) , 10.1038/NRD1551
Joel J. Bergh, Hung-Yun Lin, Lawrence Lansing, Seema N. Mohamed, Faith B. Davis, Shaker Mousa, Paul J. Davis, Integrin αVβ3 Contains a Cell Surface Receptor Site for Thyroid Hormone that Is Linked to Activation of Mitogen-Activated Protein Kinase and Induction of Angiogenesis Endocrinology. ,vol. 146, pp. 2864- 2871 ,(2005) , 10.1210/EN.2005-0102
Toshie Fujishima, Genichiro Tsuji, Chika Tanaka, Hiroshi Harayama, Novel vitamin D receptor ligands having a carboxyl group as an anchor to arginine 274 in the ligand-binding domain. The Journal of Steroid Biochemistry and Molecular Biology. ,vol. 121, pp. 60- 62 ,(2010) , 10.1016/J.JSBMB.2010.04.020
Manuel Tardáguila, Elena González-Gugel, Aurora Sánchez-Pacheco, Aurora kinase B activity is modulated by thyroid hormone during transcriptional activation of pituitary genes Molecular Endocrinology. ,vol. 25, pp. 385- 393 ,(2011) , 10.1210/ME.2010-0446