A NOVEL SYNTHESIS OF 2,3-DIHYDRO[1,5]BENZOTHIAZEPIN-4(5H)-ONES
作者： Jean-Charles Lancelot , Bertrand Letois , Carmela Saturnono , Paolo De Caprariis , Max Robba
DOI: 10.1080/00304949209355701
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摘要:
core.ac.uk
sci-hub.se 参考文章(9)
Sachio Ohno, Kihachiro Izumi, Kiyoshi Mizukoshi, Kazuo Kato, Mikio Hori, Synthesis of a new potent anti-ulcer and gastric secretory inhibiting agent, (-)-cis-2,3-dihidro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5-benzothiazepin-4(5H)-one hydrochloride(BTM-1086), and related compounds. Chemical & Pharmaceutical Bulletin. ,vol. 31, pp. 1780- 1783 ,(1983) , 10.1248/CPB.31.1780
MARI SAKUMA, MASAYOSHI YOSHIKAWA, YOSHISHIGE SATO, The whole body autoradiographic studies on the distribution of 14 C-labeled new 1,5-benzothiazepine derivative ( 14 C-CRD-401) in mice. Chemical & Pharmaceutical Bulletin. ,vol. 19, pp. 995- 1005 ,(1971) , 10.1248/CPB.19.995
Mohammed A. Matlib, Shin-Woong Lee, Alain Depover, Arnold Schwartz, A specific inhibitory action of certain benzothiazepines and benzodiazepines on the sodium-calcium exchange process of heart and brain mitochondria European Journal of Pharmacology. ,vol. 89, pp. 327- 328 ,(1983) , 10.1016/0014-2999(83)90518-6
TAKU NAGAO, MASANORI SATO, HIROMICHI NAKAJIMA, AKIO KIYOMOTO, Studies on a new 1,5-benzothiazepine derivative (CRD-401). IV. Coronary vasodilating effect and structure-activity relationship. Chemical & Pharmaceutical Bulletin. ,vol. 21, pp. 92- 97 ,(1973) , 10.1248/CPB.21.92
HIROSHI KUGITA, HIROZUMI INOUE, MUNEYOSHI IKEZAKI, SATOSHI TAKEO, Synthesis of 1, 5-Benzothiazepine Derivatives. I Chemical & Pharmaceutical Bulletin. ,vol. 18, pp. 2028- 2037 ,(1970) , 10.1248/CPB.18.2028
William J. Raich, Cliff S. Hamilton, 6-Phenylthieno[2,3-b]pyridine from 2-Nitro-3-thenaldehyde Journal of the American Chemical Society. ,vol. 79, pp. 3800- 3804 ,(1957) , 10.1021/JA01571A048
TOMIKI HASHIYAMA, AKISHIGE WATANABE, HIROZUMI INOUE, MIKIHIKO KONDA, MIKIO TAKEDA, SAKAE MURATA, TAKU NAGAO, Reactions of 3-phenylglycidic esters. V: Reaction of methyl 3-(4-methoxyphenyl)glycidate with 2-nitroaniline and synthesis of 1,5-benzodiazepine derivatives Chemical & Pharmaceutical Bulletin. ,vol. 33, pp. 2348- 2358 ,(1985) , 10.1248/CPB.33.634
John Krapcho, Ervin R. Spitzmiller, Chester F. Turk, SUBSTITUTED 2,3-DIHYDRO-1,5-BENZOTHIAZEPIN-4(5H)-ONES AND 3,4-DIHYDRO-2-PHENYL-(2H)-1,6-BENZOTHIAZOCIN-5(6H)-ONES. Journal of Medicinal Chemistry. ,vol. 6, pp. 544- 546 ,(1963) , 10.1021/JM00341A017
MICHIHIKO MIYAZAKI, TAKEO IWAKUMA, TADASU TANAKA, Synthesis of the metabolites and related compounds of Diltiazem. CHEMICAL & PHARMACEUTICAL BULLETIN. ,vol. 26, pp. 2889- 2893 ,(1978) , 10.1248/CPB.26.2889