An alternative way to analogues of avenanthramides and their antiradical activity
作者： Inese Mierina , Agnese Stikute , Anatoly Mishnev , Mara Jure
DOI: 10.1007/S00706-018-2288-6
关键词:
摘要: The paper is devoted to the synthesis of arylidene malonic acid monoanilides and cinnamoyl anilines by condensation with aromatic aldehydes. presented synthetic route applies simple, cheap, commercially available aldehydes amines, thus overcoming traditional schemes, which involve derivatives hydroxycinnamic acids. Besides, a mild effective pyridine-mediated decarboxylation carboxylic group at Csp2 in leading presented. structures obtained selected were approved additionally X-ray analysis. antiradical properties (2,2-diphenyl-1-picrylhydrazyl galvinoxyl tests) structure–activity relationships synthesized compounds studied.
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sci-hub.se 参考文章(59)
M. V. Ramana Reddy, E. Premkumar Reddy, Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof ,(2003)
Ljubomir Isakovic, Franck Raeppel, Stephane Raeppel, Arkadii Vaisburg, Amal Wahhab, Stephen William Claridge, Lijie Zhan, Naomy Bernstein, Frederic Gaudette, Marie-Claude Granger, Michael Mannion, Robert Deziel, Oscar Mario Saavedra, Nancy Zhou, Inhibitors of vegf receptor and hgf receptor signaling ,(2006)
Jae-Chul Jung, Sohyeon Moon, Dongguk Min, Woo Kyu Park, Mankil Jung, Seikwan Oh, Synthesis and Evaluation of a Series of 3,4,5-Trimethoxycinnamic Acid Derivatives as Potential Antinarcotic Agents Chemical Biology & Drug Design. ,vol. 81, pp. 389- 398 ,(2013) , 10.1111/CBDD.12087
V. I. Akhmedzhanova, I. A. Bessonova, S. Yu. Yunusov, Alkaloids of Haplophyllum perforatum Chemistry of Natural Compounds. ,vol. 12, pp. 282- 288 ,(1976) , 10.1007/BF00567798
Bruce C. Hamper, Allen S. Kesselring, Robert C. Chott, Shengtian Yang, Parallel solid-phase synthesis and high-throughput 1H NMR evaluation of a 96-member 1,2,4-trisubstituted-pyrimidin-6-one-5-carboxylic acid library. ACS Combinatorial Science. ,vol. 11, pp. 469- 480 ,(2009) , 10.1021/CC900010V
Fatemeh Tamaddon, Fatemeh Aboee, Alireza Nasiri, ZnO nanofluid as a structure base catalyst for chemoselective amidation of aliphatic carboxylic acids Catalysis Communications. ,vol. 16, pp. 194- 197 ,(2011) , 10.1016/J.CATCOM.2011.09.023
Maria C. Burla, Rocco Caliandro, Mercedes Camalli, Benedetta Carrozzini, Giovanni L. Cascarano, Liberato De Caro, Carmelo Giacovazzo, Giampiero Polidori, Riccardo Spagna, SIR2004: an improved tool for crystal structure determination and refinement Journal of Applied Crystallography. ,vol. 38, pp. 381- 388 ,(2005) , 10.1107/S002188980403225X
Hugo E. Gottlieb, Vadim Kotlyar, Abraham Nudelman, NMR Chemical Shifts of Common Laboratory Solvents as Trace Impurities. Journal of Organic Chemistry. ,vol. 62, pp. 7512- 7515 ,(1997) , 10.1021/JO971176V
G. V. Kryshtal, E. P. Serebryakov, Regio- and stereoselectivity in the addition reactions of CH-acids to aldehydes under the conditions of phase-transfer catalysis Russian Chemical Bulletin. ,vol. 44, pp. 1785- 1804 ,(1995) , 10.1007/BF00707200
Slobodan V. Jovanovic, Mihajilo Tosic, Michael G. Simic, Use of the Hammett correlation and .delta.+ for calculation of one-electron redox potentials of antioxidants The Journal of Physical Chemistry. ,vol. 95, pp. 10824- 10827 ,(1991) , 10.1021/J100179A054