Potent parp inhibitors

作者: Philip J. Hajduk , Thomas D. Penning , Sheela A. Thomas , Daryl R. Sauer , Kathy Sarris

DOI:

关键词:

摘要: The present invention relates to 1H-benzimidazole-4-carboxamides of formula (I), their preparation, and use as inhibitors the enzyme poly(ADP-ribose)polymerase for preparation drugs.

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