Efficient Synthesis of 2‐Fluoromethylated Quinolines via Copper‐Catalyzed Alkynylation and Cyclization of Fluorinated Imidoyl Iodides
作者： Shan Li , Yafen Yuan , Jiangtao Zhu , Haibo Xie , Zixian Chen
关键词:
摘要: 2-Fluoromethylated quinolines were synthesized through the reaction of N-aryl-fluorinated imidoyl iodides with terminal alkynes in good yields by catalysis copper(I) iodide (CuI) alone.
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