Die identifisering van fenielbottersuur aromatiese metaboliete in die urien van die blou-aap

Mietha M. Van der Walt , Gisella Terre'Blanche , Jacobus J. Bergh , Lodewyk J. Mienie
Suid-Afrikaans Tydskrif vir Natuurwetenskap en Tegnologie / <i>South African Journal of Science and Technology</i> 37 ( 1) 10 -14

2018
Imidazo[1,2-α]pyridines possess adenosine A1 receptor affinity for the potential treatment of cognition in neurological disorders

Roslyn Lefin , Mietha M. van der Walt , Pieter J. Milne , Gisella Terre'Blanche
Bioorganic & Medicinal Chemistry Letters 27 ( 17) 3963 -3967

7
2017
C2-substituted quinazolinone derivatives exhibit A1 and/or A2A adenosine receptor affinities in the low micromolar range.

Lianie Pieterse , Mietha M. van der Walt , Gisella Terre'Blanche
Bioorganic & Medicinal Chemistry Letters 30 ( 16) 127274

2020
Treatment of an adrenomyeloneuropathy patient with Lorenzo's oil and supplementation with docosahexaenoic acid-A case report

Gisella Terre'Blanche , Mietha M van der Walt , Jacobus J Bergh , Lodewyk J Mienie
Lipids in Health and Disease 10 ( 1) 152 -152

10
2011
Synthesis and evaluation of methoxy substituted 2-benzoyl-1-benzofuran derivatives as lead compounds for the development adenosine A1 and/or A2A receptor antagonists.

Helena D. Janse van Rensburg , Lesetja J. Legoabe , Gisella Terre'Blanche , Janine Aucamp
Bioorganic Chemistry 94 103459

3
2020
Benzopyrone represents a privilege scaffold to identify novel adenosine A1/A2A receptor antagonists.

Mietha M. van der Walt , Gisella Terre'Blanche
Bioorganic Chemistry 77 136 -143

3
2018
Screening of novel pentacyclo-undecylamines for neuroprotective activity.

Werner J Geldenhuys , Gisella Terre'Blanche , Cornelis J Van der Schyf , Sarel F Malan
European Journal of Pharmacology 458 ( 1) 73 -79

33
2003
Neurotoxicity studies with the monoamine oxidase B substrate 1-methyl-3-phenyl-3-pyrroline.

Modupe O. Ogunrombi , Sarel F. Malan , Gisella Terre'Blanche , Kay Castagnoli
Life Sciences 81 ( 6) 458 -467

9
2007
Physicochemical prediction of a brain–blood distribution profile in polycyclic amines

Jaco Zah , Gisella Terre'Blanche , Elardus Erasmus , Sarel F. Malan
Bioorganic & Medicinal Chemistry 11 ( 17) 3569 -3578

40
2003
Methoxy substituted 2-benzylidene-1-indanone derivatives as A1 and/or A2A AR antagonists for the potential treatment of neurological conditions

Helena D. Janse van Rensburg , Lesetja J. Legoabe , Gisella Terre'Blanche , Mietha M. Van der Walt
MedChemComm 10 ( 2) 300 -309

5
2019
8-(3-phenylpropyl)-1,3,7-triethylxanthine is a synthetic caffeine substitute with stronger metabolic modulator activity.

David F. Carrageta , Tânia R. Dias , Ivana Jarak , Marco G. Alves
Toxicology in Vitro 53 114 -120

2
2018
Evaluation of 2‐benzylidene‐1‐tetralone derivatives as antagonists of A1 and A2A adenosine receptors

Lesetja J. Legoabe , Mietha M. Van der Walt , Gisella Terre'Blanche
Chemical Biology & Drug Design 91 ( 1) 234 -244

8
2018
Design, synthesis and evaluation of amino-3, 5-dicyanopyryridines and thieno [2, 3-b] pyridines as ligands of adenosine receptors

Gaofenngwe Nkomba , Gisella Terre'Blanche , Helena Dorathea Janse van Rensburg , Lesetja J Legoabe

2022
5-Substituted 2-benzylidene-1-tetralone analogues as A 1 and/or A 2A antagonists for the potential treatment of neurological conditions

H.D. Janse van Rensburg , G. Terre'Blanche , M.M. van der Walt , L.J. Legoabe
Bioorganic Chemistry 74 251 -259

7
2017
Selected C8 two-chain linkers enhance the adenosine A1/A2A receptor affinity and selectivity of caffeine.

M.M. van der Walt , G. Terre'Blanche
European Journal of Medicinal Chemistry 125 652 -656

17
2017
Investigating the potential neuroprotective effects of statins on DNA damage in mouse striatum.

T.N. Coetsee , P.J. Pretorius , G. Terre’Blanche , J.J. Bergh
Food and Chemical Toxicology 46 ( 9) 3186 -3192

7
2008
Therapeutic potentials of agonist and antagonist of adenosine receptors in type 2 diabetes

Olakunle Sanni , G Terre’Blanche
Reviews in Endocrine and Metabolic Disorders 22 ( 4) 1073 -1090

12
2021
2022
Synthesis and Structure Activity Relationships of Chalcone based Benzocycloalkanone Derivatives as Adenosine A1 and/or A2A Receptor Antagonists.

Helena D. Janse van Rensburg , Lesetja J. Legoabe , Gisella Terre’Blanche
Drug Research 70 ( 06) 243 -256

2020