Harnessing the power of transition metals in solid-phase peptide synthesis and key steps in the (semi)synthesis of proteins.

Ashraf Brik , Shay Laps , Gandhesiri Satish
Chemical Society Reviews 50 ( 4) 2367 -2387

1
2021
Enhanced Live-Cell Delivery of Synthetic Proteins Assisted by Cell-Penetrating Peptides Fused to DABCYL.

Ashraf Brik , Guy Mann , Gandhesiri Satish , Shaswati Mandal
Angewandte Chemie 60 ( 13) 7333 -7343

26
2021
Chemical Synthesis of Ubiquitinated Proteins for Biochemical Studies

Ashraf Brik , Ganga B. Vamisetti , Gandhesiri Satish
Total Chemical Synthesis of Proteins 383 -410

2021
Palladium-Mediated Cleavage of Proteins with Thiazolidine-Modified Backbone in Live Cells.

Guy Mann , Gandhesiri Satish , Roman Meledin , Ganga B. Vamisetti
Angewandte Chemie 58 ( 38) 13540 -13549

12
2019
Nickel-Catalyzed Annulation of 2′-Aminochalcones: A Simplistic Access to 4-Styryl and 2,4-Distyrylquinolines

Gandhesiri Satish , Polu Ashok , Laxman Kota , Andivelu Ilangovan
ChemistrySelect 4 ( 4) 1346 -1349

4
2019
Direct Amidation of 2′-Aminoacetophenones Using I2-TBHP: A Unimolecular Domino Approach toward Isatin and Iodoisatin

Andivelu Ilangovan , Gandhesiri Satish
Journal of Organic Chemistry 79 ( 11) 4984 -4991

54
2014
Copper-catalyzed oxidative amination of methanol to access quinazolines

Gandhesiri Satish , Ashok Polu , Laxman Kota , Andivelu Ilangovan
Organic and Biomolecular Chemistry 17 ( 19) 4774 -4782

7
2019
Iodine-Mediated C–H Functionalization of sp, sp2, and sp3 Carbon: A Unified Multisubstrate Domino Approach for Isatin Synthesis

Gandhesiri Satish , Ashok Polu , Thangeswaran Ramar , Andivelu Ilangovan
Journal of Organic Chemistry 80 ( 10) 5167 -5175

47
2015
On-Demand Detachment of Succinimides on Cysteine to Facilitate (Semi)Synthesis of Challenging Proteins.

Ganga B. Vamisetti , Gandhesiri Satish , Prasad Sulkshane , Guy Mann
Journal of the American Chemical Society 142 ( 46) 19558 -19569

3
2020
K2S2O8-mediated metal-free direct C–H functionalization of quinones using arylboronic acids

Andivelu Ilangovan , Ashok Polu , Gandhesiri Satish
Organic chemistry frontiers 2 ( 12) 1616 -1620

34
2015
Copper-mediated selective C-H activation and cross-dehydrogenative C-N coupling of 2'-aminoacetophenones

Andivelu Ilangovan , Gandhesiri Satish
Organic Letters 15 ( 22) 5726 -5729

52
2013
Iodine/TBHP

Gandhesiri Satish
Synlett 26 ( 13) 1913 -1914

2015
A short binding site in the KPC1 ubiquitin ligase mediates processing of NF-κB1 p105 to p50: A potential for a tumor-suppressive PROTAC

Gilad Goldhirsh , Yelena Kravtsova-Ivantsiv , Gandhesiri Satish , Tamar Ziv
Proceedings of the National Academy of Sciences 118 ( 49) e2117254118 -e2117254118

7
2021
Synthesis and delivery of a stable phosphorylated ubiquitin probe to study ubiquitin conjugation in mitophagy

Guy Mann , Gandhesiri Satish , Prasad Sulkshane , Shaswati Mandal
Chemical Communications 57 ( 74) 9438 -9441

16
2021
Single-shot flow synthesis of d-proteins for mirror-image phage display

Alex J Callahan , Satish Gandhesiri , Tara L Travaline , Lia Lozano Salazar
Smpte Journal

2023
Synthesis and Evaluation of Ubiquitin--Dioxetane Conjugate as a Chemiluminescent Probe for Monitoring Deubiquitinase Activity

Sara Gutkin , Satish Gandhesiri , Ashraf Brik , Doron Shabat
Bioconjugate Chemistry 32 ( 10) 2141 -2147

7
2021
Mirror-image ligand discovery enabled by single-shot fast-flow synthesis of D-proteins

Alex J Callahan , Satish Gandhesiri , Tara L Travaline , Rahi M Reja
Nature Communications 15 ( 1) 1813 -1813

4
2024
Automated flow peptide synthesis enables engineering of proteins with stabilized transient binding pockets

Anna Charalampidou , Thomas Nehls , Christian Meyners , Satish Gandhesiri
ACS Central Science 10 ( 3) 649 -657

1
2024
Equimolar Cross-Coupling Using Reactive Coiled Coils for Stable Covalent Protein Assemblies

Hironori Takeuchi , Elee Shimshoni , Satish Gandhesiri , Andrei Loas

2024