Occupancy of Dopamine D2 and D3 Receptors by a Novel D3 Partial Agonist BP1. 4979: A [11C]-(+)-PHNO PET Study in Humans
Bernard Le Foll , Patricia Di Ciano , Esmaeil Mansouri , Alan A Wilson
NEUROPSYCHOPHARMACOLOGY 43 S453 -S454
2017
TETRAHEDRON: ASYMMETRY REPORT NUMBER 59
OB Sutcliffe , MR Bryce , GJA Conceiçao , PJS Moran
Tetrahedron: Asymmetry 14 ( 16)
Anxiogenic effects of CCK agonists in a nonhuman primate model: Central or peripheral
RM Palmour , C Durieux , BP Roques , P Bertrand
CCK 93 19 -22
9
1993
Preparation of 1-bis (aryl) methyl-3-(alkylsulfonyl) arylmethyleneazetidines as cannabinoid CB1 receptor antagonists
S Mignani , O Hittinger , D Archard , H Bouchard
Chemical Abstracts. France: Aventis Pharma SA 236982s -236982s
8
2000
From Random Screening of Chemical Libraries to the Optimization of FPP-Competitive Inhibitors of Farnesyltransferase
Alain Commerçon , Jean-Dominique Bourzat , Jacques Lavayre , Clive Brealey
Humana Press 115 -144
2001
Novel arylpiperazine derivatives
Marcel Morvan , Jeanne-Marie Lecomte , Marc Capet , Isabelle Berrebi-Bertrand
2008
N-phenyl n-acetamido glycinamides, leur preparation et les medicaments les contenant
Franco Manfre , Jean-Dominique Bourzat , Claude Cotrel , Claude Guyon
1991
Derives de glycinamide, leur preparation et les medicaments les contenant
Franco Manfre , Jean-Dominique Bourzat , Claude Cotrel , Claude Guyon
1991
Derives de n-phenyl glycinamide, leur preparation et les medicaments les contenant
Franco Manfre , Jean-Dominique Bourzat , Claude Cotrel , Claude Guyon
1991
N-phenyl n-alcoxycarbonylalkyle glycinamides, leur preparation et les medicaments les contenant
Franco Manfre , Claude Cotrel , Claude Guyon , Gerard Roussel
1991
Histamine and tele-methylhistamine quantification in cerebrospinal fluid from narcoleptic subjects by liquid chromatography tandem mass spectrometry with precolumn derivatization.
Mikaël Croyal , Yves Dauvilliers , Olivier Labeeuw , Marc Capet
Analytical Biochemistry 409 ( 1) 28 -36
33
2011
Determination of the binding mode and interacting amino-acids for dibasic H3 receptor antagonists
Olivia Poupardin-Olivier , Isabelle Berrebi-Bertrand , Jeanne-Marie Lecomte , Jean-Charles Schwartz
Bioorganic & Medicinal Chemistry 21 ( 15) 4526 -4529
13
2013
Synthesis and evaluation of amides surrogates of dopamine D3 receptor ligands.
Mickaël Jean , Jacques Renault , Nicolas Levoin , Denis Danvy
Bioorganic & Medicinal Chemistry Letters 20 ( 18) 5376 -5379
5
2010
Novel and highly potent histamine H3 receptor ligands. Part 1: withdrawing of hERG activity
Nicolas Levoin , Olivier Labeeuw , Thierry Calmels , Olivia Poupardin-Olivier
Bioorganic & Medicinal Chemistry Letters 21 ( 18) 5378 -5383
13
2011
Novel and highly potent histamine H3 receptor ligands. Part 2: Exploring the cyclohexylamine-based series
Olivier Labeeuw , Nicolas Levoin , Olivia Poupardin-Olivier , Thierry Calmels
Bioorganic & Medicinal Chemistry Letters 21 ( 18) 5384 -5388
9
2011
Refined docking as a valuable tool for lead optimization: application to histamine H3 receptor antagonists.
Nicolas Levoin , Thierry Calmels , Olivia Poupardin-Olivier , Olivier Labeeuw
Archiv Der Pharmazie 341 ( 10) 610 -623
35
2008
Synthesis and evaluation of a 2-benzothiazolylphenylmethyl ether class of histamine H4 receptor antagonists.
Olivier Labeeuw , Nicolas Levoin , Xavier Billot , Denis Danvy
Bioorganic & Medicinal Chemistry Letters 26 ( 21) 5263 -5266
5
2016
Improving selectivity of dopamine D3 receptor ligands.
Marc Capet , Thierry Calmels , Nicolas Levoin , Denis Danvy
Bioorganic & Medicinal Chemistry Letters 26 ( 3) 885 -888
7
2016
Congo red protects against toxicity of β-amyloid peptides on rat hippocampal neurones
Marie-Claude Burgevin , Marylène Passat , Nadine Daniel , Marc Capet
Neuroreport 5 ( 18) 2429 -2432
39
1994
Novel and highly potent histamine H3 receptor ligands. Part 3: an alcohol function to improve the pharmacokinetic profile.
Marc Capet , Olivier Labeeuw , Nicolas Levoin , Olivia Poupardin-Olivier
Bioorganic & Medicinal Chemistry Letters 23 ( 9) 2548 -2554
4
2013