Direct photocapture of bromodomains using tropolone chemical probes

作者: Erik C. Hett , Eugene L. Piatnitski Chekler , Arindrajit Basak , Paul D. Bonin , R. Aldrin Denny

DOI: 10.1039/C5MD00070J

关键词: TropoloneBRD4TroponeTubulinProteomeStereochemistryCombinatorial chemistryLysineChemistryBET inhibitorBromodomain

摘要: Tropolone probes directly photoaffinity label bromodomains.

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