Antiviral, highly water soluble, stable, crystalline salts of 2′, 3′-dideoxyinosine, 2′, 3′-dideoxy-2′, 3′-didehydrothymidine and 2′, 3′-dideoxy-2′-fluoroinosine

作者: Robert K. Perrone , Murray A. Kaplan , Joseph B. Bogardus

DOI:

关键词: Water soluble2'3' dideoxyinosineStereochemistryChemistryOrganic chemistry

摘要: Provided are very highly water soluble, stable, crystalline salts of 2′,3′-dideoxy-2′,3′-didehydrothymidine (“d4T”), 2′,3′-dideoxyinosine (“ddI”), and 2′,3′-dideoxy-2′-fluoroinosine (“F-ddI”). Such useful as intermediates or antiviral agents.

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