Regiospecific Synthesis of Certain 1,2,3,4-Tetrasubstituted Benzenes in One Step via a Benzene Cyclization
作者： Lawrence E. Fisher , Joan M. Caroon
DOI: 10.1080/00397918908050974
关键词: Aniline 、 Organic chemistry 、 Chemistry 、 One-Step 、 Benzene 、 Single step 、 Electrophile
摘要: Abstract Tetrasubstituted benzenes of type 3 are obtained regiospecifically in a single step by the treatment 1-fluoro-4-methoxy-5-carbo-tert-butoxy aniline with tert-butyllithium followed reaction an electrophile.
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