Methods and use of bifunctional enzyme-building clamp-shaped molecules

作者: Alan Berezov , Zheng Cai , Hongtao Zhang , Mark I. Greene

DOI:

关键词: ClampBiochemistryPhosphofructokinase 2Cancer therapyCellMoleculeChemistry

摘要: This invention is in the fields of cancer therapy. More particularly it concerns compounds which are useful agents for inhibiting cell proliferative disorders, especially those disorders characterized by over activity and/or inappropriate a EGFR, including EGFR-related cancers, and methods treating these disorders.

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