Process for making fingolimod

作者: Jozef Krajcovic , Reinerus Gerardus Gieling

DOI:

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摘要: The invention relates to a process of making fingolimod formula (1), or an acid addition salt thereof comprising step reacting the compound (11) and/or (14) thereof, in solvent with hydrogen presence hydrogenation catalyst, preferably palladium and optionally converting (1) into salt, compounds (14), processes them their use fingolimod.

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