D-Tyr—Ser—Gly—Phe—Leu—Thr, a highly preferential ligand for δ-opiate receptors

作者: Gilles Gacel , Marie-Claude Fournie-Zaluski , Bernard P. Roques

DOI: 10.1016/0014-5793(80)80229-8

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参考文章(15)
P Cuatrecasas, K J Chang, Multiple opiate receptors. Enkephalins and morphine bind to receptors of different specificity. Journal of Biological Chemistry. ,vol. 254, pp. 2610- 2618 ,(1979) , 10.1016/S0021-9258(17)30115-1
Rüdiger Schulz, Michael Wüster, Heinz Krenss, Albert Herz, Selective development of tolerance without dependence in multiple opiate receptors of mouse vas deferens Nature. ,vol. 285, pp. 242- 243 ,(1980) , 10.1038/285242A0
Henk Rigter, Tracy J. Hanna, Rita B. Messing, Joe L. Martinez, Beatriz J. Vasquez, Robert A. Jensen, John Veliquette, James L. McGaugh, Enkephalins interfere with acquisition of an active avoidance response Life Sciences. ,vol. 26, pp. 337- 345 ,(1980) , 10.1016/0024-3205(80)90149-6
H.W. KOSTERLITZ, J.A.H. LORD, S.J. PATERSON, ANGELA A. WATERFIELD, Effects of changes in the structure of enkephalins and of narcotic analgesic drugs on their interactions with μ and δ-receptors British Journal of Pharmacology. ,vol. 68, pp. 333- 342 ,(1980) , 10.1111/J.1476-5381.1980.TB10422.X
Bernard P. Roques, Gilles Gacel, Marie-Claude Fournie-Zaluski, Bernard Senault, Jeanne-Marie Lecomte, Demonstration of the crucial role of the phenylalanine moiety in enkephalin analogues for differential recognition of the μ- and δ-receptors European Journal of Pharmacology. ,vol. 60, pp. 109- 110 ,(1979) , 10.1016/0014-2999(79)90059-1
J. R. Smith, E. J. Simon, Selective protection of stereospecific enkephalin and opiate binding against inactivation by N-ethylmaleimide: evidence for two classes of opiate receptors. Proceedings of the National Academy of Sciences of the United States of America. ,vol. 77, pp. 281- 284 ,(1980) , 10.1073/PNAS.77.1.281
C. Garbay-Jaureguiberry, B.P. Roques, R. Oberlin, 1H and 13C NMR studies of conformational behaviour of Leu-enkephalin FEBS Letters. ,vol. 76, pp. 93- 98 ,(1977) , 10.1016/0014-5793(77)80128-2
C. Garbay-Jaureguiberry, B.P. Roques, R. Oberlin, M. Anteunis, A.K. Lala, Preferential conformation of the endogenous opiate-like pentapeptide met-enkephalin in DMSO-d6 solution determined by high field 1H NMR Biochemical and Biophysical Research Communications. ,vol. 71, pp. 558- 565 ,(1976) , 10.1016/0006-291X(76)90823-8
J. F. Kachur, R. J. Miller, M. Field, Control of guinea pig intestinal electrolyte secretion by a delta-opiate receptor. Proceedings of the National Academy of Sciences of the United States of America. ,vol. 77, pp. 2753- 2756 ,(1980) , 10.1073/PNAS.77.5.2753
B. MALFROY, J. P. SWERTS, A. GUYON, B. P. ROQUES, J. C. SCHWARTZ, High-affinity enkephalin-degrading peptidase in brain is increased after morphine Nature. ,vol. 276, pp. 523- 526 ,(1978) , 10.1038/276523A0