An expeditious approach to tri-substituted chiral thiazolines
作者： Raid J Abdel-Jalil , Muhammad Saeed , Wolfgang Voelter
DOI: 10.1016/S0040-4039(01)00188-5
关键词:
摘要: A regio- and stereoselective route from the cis-oriented epoxytriflate pentoses 1 4 via 4-amino-4-deoxy sugars 2 5 to chiral thiazoline derivatives 3a–e 6a–e in high yields is described.
elsevier.com
sci-hub.se 参考文章(13)
Raid J. Abdel-Jalil, Raed A. Al-Qawasmeh, Yousef Al-Abed, Wolfgang Voelter, A stereospecific synthesis of tetra-substituted chiral piperazines Tetrahedron Letters. ,vol. 39, pp. 7703- 7704 ,(1998) , 10.1016/S0040-4039(98)01677-3
Akira Ino, Yasushi Hasegawa, Akira Murabayashi, Synthetic studies of thiazoline and thiazolidine-containing natural products — 2. Total synthesis of the antimycoplasma antibiotic micacocidin Tetrahedron. ,vol. 55, pp. 10283- 10294 ,(1999) , 10.1016/S0040-4020(99)00583-9
Spencer Knapp, David Vocadlo, Zhinong Gao, Brian Kirk, Jianping Lou, Stephen G. Withers, NAG-thiazoline, An N-Acetyl-β-hexosaminidase Inhibitor That Implicates Acetamido Participation Journal of the American Chemical Society. ,vol. 118, pp. 6804- 6805 ,(1996) , 10.1021/JA960826U
Heinz-Werner Hagedorn, Hans Merten, Reinhard Brossmer, Synthesis of the deculopyranosonic acid analog of N-acetylneuraminic acid, its 5-epimer and 6-epimer, and of 5-acetamido-1,3,5-trideoxy-d-glycero-d-galactonon-2-ulopyranose☆ Carbohydrate Research. ,vol. 236, pp. 89- 96 ,(1992) , 10.1016/0008-6215(92)85008-N
Raymond J. Bergeron, Jan Wiegand, John B. Dionis, Majia Egli-Karmakka, Joerg Frei, Alica Huxley-Tencer, Heinrich H. Peter, Evaluation of desferrithiocin and its synthetic analogues as orally effective iron chelators. Journal of Medicinal Chemistry. ,vol. 34, pp. 2072- 2078 ,(1991) , 10.1021/JM00111A023
Raed A. Al-Qawasmeh, Raid J. Abdel-Jalil, Taleb H. Al-Tel, René Thürmer, Wolfgang Voelter, A useful regioselective approach to episulfides via cis-oriented anhydro triflate sugars Tetrahedron Letters. ,vol. 39, pp. 8257- 8258 ,(1998) , 10.1016/S0040-4039(98)01885-1
Christopher D.J. Boden, Mark C Norley, Gerald Pattenden, Total synthesis of the thiazoline-based cyclopeptide cyclodidemnamide Tetrahedron Letters. ,vol. 37, pp. 9111- 9114 ,(1996) , 10.1016/S0040-4039(96)02099-0
Michael Z. Hoemann, Konstantinos A. Agrios, Jeffrey Aubé, TOTAL SYNTHESIS OF (+)-CURACIN A, A MARINE CYTOTOXIC AGENT Tetrahedron. ,vol. 53, pp. 11087- 11098 ,(1997) , 10.1016/S0040-4020(97)00368-2
R. Thurmer, R.J. Abdel-Jalil, R.A. Al-Qawasmeh, T.H. Al-Tel, W. Voelter, Y. Al-Abed, Epoxy Pyranoses, Chiral Synthons for Versatile Regio- and Stereocontrolled Functionalizations Polish Journal of Chemistry. ,vol. 73, pp. 55- 69 ,(1999)
Gaik B. Kok, Michael Campbell, Brendan Mackey, Mark von Itzstein, Synthesis and biological evaluation of sulfur isosters of the potent influenza virus sialidase inhibitors 4-amino-4-deoxy- and 4-deoxy-4-guanidino-Neu5Ac2en Journal of The Chemical Society-perkin Transactions 1. pp. 2811- 2815 ,(1996) , 10.1039/P19960002811