Protein kinase C-α inhibitors; structure-activity relationships in bis-indole series
作者： Guojian Xie , Jürg Zimmermann , Thomas Meyer , J. William Lown
DOI: 10.1016/0960-894X(95)00060-7
关键词:
摘要: Abstract To assess the role of amine and ester containing oligopeptide side-chains in bis-indole protein kinase C inhibitors, six novel hybrids this series were synthesized. These new compounds displayed effective inhibitory activity against C-α.
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