Aminium salts of 1,2,3-triazoles as prodrugs of drugs including antiviral agents

作者: Alicia Regueiro-Ren , John F. Kadow

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摘要: This disclosure provides compounds having drug and bio-affecting properties, their pharmaceutical compositions method of use. In particular, the is concerned with new aminium salts 1,2,3-triazoles which can be used as prodrugs to improve solubility or properties 1,2,3-triazole containing compounds. More particularly, present relates N-aminium-1,2,3-triazoles that are useful antiviral agents specifically for treatment HIV AIDS.

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