SD0006: a potent, selective and orally available inhibitor of p38 kinase.
作者： Barry L. Burnette , Shaun Selness , Raj Devraj , Gail Jungbluth , Ravi Kurumbail
DOI: 10.1159/000227286
关键词:
摘要: SD0006 is a diarylpyrazole that was prepared as an inhibitor of p38 kinase-α (p38α). In vitro, selective for p38α kinase over 50 other kinases screened (including p38γ and p38δ with modest
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