One-pot synthesis of benzofused heteroaryl azoles via tandem C-heteroatom coupling/C–H activation of azoles

作者: Xurong Qin , Xuefeng Cong , Dongbing Zhao , Jingsong You , Jingbo Lan

DOI: 10.1039/C1CC10572H

关键词:

摘要: The Cu(I) or Pd(II)-catalyzed cross-couplings of gem-dihaloolefins with azoles via tandem C-heteroatom coupling/C–H activation for the preparation benzofused heteroaryl have been developed.

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