Substituted 3 - (thiazole - 4 - carbonyl) - or 3 - (thiazole - 2 - carbonyl) aminopropionic acid derivatives and their use as pharmaceuticals
作者： Georg Horstick , Klaus Wirth , Christian Buning , Josef Pernerstorfer , Sven Ruf
DOI:
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摘要: The present invention relates to compounds of the formulae (Ia) and (Ib), wherein G, R 10 , 30 40 50 60 have meanings indicated in claims, which are valuable pharmaceutical active compounds. They inhibitors protease cathepsin A, useful for treatment diseases such as atherosclerosis, heart failure, renal diseases, liver or inflammatory example. furthermore processes preparation la lb, their use compositions comprising them.
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