Amino acids in the syntheses of heterocyclic systems: Syntheses and radiostability of novel biologically active triazoles containing the sulfonamide moiety

作者: A. M. Sh. El-Sharief , M. M. Ghorab , M. S. A. El-Gaby , Sh. I. Mohamed , Y. A. Ammar

DOI: 10.1002/HC.10037

关键词:

摘要: A number of novel triazoles 2a–f, 4, 9, 10, 12, 15; triazolothiadiazoles 6, 8, 11, 16; triazolothiadiazine 5; and triazolotriazine 14 were synthesized characterized by elemental analyses spectral data. Six the compounds showed antifungal activity compared with fungicide Mycostatine. Radiosterilization biologically active 9b, 10 in dry state may prove to be applicable at sterile dose 25 kGy. © 2002 Wiley Periodicals, Inc. Heteroatom Chem 13:316–323, 2002; Published online Interscience (www.interscience.wiley.com). DOI 10.1002/hc.10037

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