Selective palladium-catalyzed aminations on dichloropyridines
作者： Tim H.M Jonckers , Bert U.W Maes , Guy L.F Lemière , Roger Dommisse
DOI: 10.1016/S0040-4020(01)00659-7
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摘要: Abstract Palladium-catalyzed amination proved to be a valuable strategy for the selective introduction of aromatic and heteroaromatic amines, including aminopyridines aminodiazines, on dichloropyridines. The use mild conditions resulted in maximum selectivity excellent base sensitive functional group tolerance.
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