Predicting Skin Permeability from Complex Chemical Mixtures: Dependency of Quantitative Structure Permeation Relationships on Biology of Skin Model Used
作者： Jim E. Riviere , James D. Brooks
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摘要: … vascularized model, which are not operative in the diffusion cell system. The pharmacokinetics of penetration through a dermatomed skin model versus an intact epidermal-dermal skin …
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Solvent systems and their selection in pharmaceutics and biopharmaceutics Springer : AAPS Press. ,(2007) , 10.1007/978-0-387-69154-1
Dermal Absorption Models in Toxicology and Pharmacology CRC Press. ,(2005) , 10.1201/9780203020821
Catarina Rosado, Sheree E. Cross, W. John Pugh, Michael S. Roberts, Jonathan Hadgraft, Effect of vehicle pretreatment on the flux, retention, and diffusion of topically applied penetrants in vitro Pharmaceutical Research. ,vol. 20, pp. 1502- 1507 ,(2003) , 10.1023/A:1025778731901
Sheree E. Cross, W. John Pugh, Jonathan Hadgraft, Michael S. Roberts, Probing the effect of vehicles on topical delivery: understanding the basic relationship between solvent and solute penetration using silicone membranes. Pharmaceutical Research. ,vol. 18, pp. 999- 1005 ,(2001) , 10.1023/A:1010996513458
Russell O. Potts, Richard H. Guy, Predicting skin permeability. Pharmaceutical Research. ,vol. 9, pp. 663- 669 ,(1992) , 10.1023/A:1015810312465
Jim E. Riviere, James D. Brooks, James L. Yeatts, Elisha L. Koivisto, Surfactant Effects on Skin Absorption of Model Organic Chemicals: Implications for Dermal Risk Assessment Studies Journal of Toxicology and Environmental Health. ,vol. 73, pp. 725- 737 ,(2010) , 10.1080/15287391003614026
Sheree E. Cross, Yuri G. Anissimov, Beatrice M. Magnusson, Michael S. Roberts, Bovine-serum-albumin-containing receptor phase better predicts transdermal absorption parameters for lipophilic compounds. Journal of Investigative Dermatology. ,vol. 120, pp. 589- 591 ,(2003) , 10.1046/J.1523-1747.2003.12083.X
Filomena Martins, Michael H. Abraham, Human Skin Permeation and Partition: General Linear Free‐Energy Relationship Analyses Journal of Pharmaceutical Sciences. ,vol. 93, pp. 1508- 1523 ,(2004) , 10.1002/JPS.20070
Sheree E. Cross, Beatrice M. Magnusson, Gareth Winckle, Yuri Anissimov, Michael S. Roberts, Determination of the effect of lipophilicity on the in vitro permeability and tissue reservoir characteristics of topically applied solutes in human skin layers Journal of Investigative Dermatology. ,vol. 120, pp. 759- 764 ,(2003) , 10.1046/J.1523-1747.2003.12131.X
SK Chang, JE Riviere, Percutaneous absorption of parathion in vitro in porcine skin: Effects of dose, temperature, humidity, and perfusate composition on absorptive flux Toxicological Sciences. ,vol. 17, pp. 494- 504 ,(1991) , 10.1016/0272-0590(91)90200-N