Synthesis and biological activity of novel 3-heteroaryl-2H-pyrido[4,3-e][1,2,4]thiadiazine and 3-heteroaryl-2H-benzo[e][1,2,4]thiadiazine 1,1-dioxides
作者： Katarzyna Gobis , Henryk Foks , Jarosłw Sławiński , Ewa Augustynowicz-Kopeć , Agnieszka Napiórkowska
DOI: 10.1007/S00706-013-0988-5
关键词:
摘要: … In an effort to develop new and effective chemotherapeutic agents for the treatment of tuberculosis, several series of heterocyclic compounds based on a sulfonamidine scaffold have …
springer.com
paperity.org参考文章(26)
Guy P. Youmans, Anne Stewart Youmans, A METHOD FOR THE DETERMINATION OF THE RATE OF GROWTH OF TUBERCLE BACILLI BY THE USE OF SMALL INOCULA1 Journal of Bacteriology. ,vol. 58, pp. 247- 255 ,(1949) , 10.1128/JB.58.2.247-255.1949
D.L. Comins, S. O’Connor, R.S. Al-awar, Pyridines and their Benzo Derivatives: Reactivity at the Ring Comprehensive Heterocyclic Chemistry III. ,vol. 7, pp. 41- 99 ,(2008) , 10.1016/B978-008044992-0.00602-7
Andrejus Korolkovas, Essentials of medicinal chemistry ,(1976)
T. C. CORBY, P. H. ELWORTHY, Identification of the site of solubilization of various compounds by cetomacrogol Journal of Pharmacy and Pharmacology. ,vol. 23, ,(2011) , 10.1111/J.2042-7158.1971.TB08768.X
Katarzyna Gobis, Henryk Foks, Jarosław Sławiński, Artur Sikorski, Damian Trzybiński, Ewa Augustynowicz-Kopeć, Agnieszka Napiórkowska, Krzysztof Bojanowski, Synthesis, structure, and biological activity of novel heterocyclic sulfonyl-carboximidamides Monatshefte Fur Chemie. ,vol. 144, pp. 647- 658 ,(2013) , 10.1007/S00706-012-0888-0
Ahmed Kamal, K. Srinivasa Reddy, S. Kaleem Ahmed, M. Naseer A. Khan, Rakesh K. Sinha, J.S. Yadav, Sudershan K. Arora, Anti-tubercular agents. Part 3. Benzothiadiazine as a novel scaffold for anti-Mycobacterium activity. Bioorganic & Medicinal Chemistry. ,vol. 14, pp. 650- 658 ,(2006) , 10.1016/J.BMC.2005.08.063
Xin Chen, Shuzhen Zhang, Yanchun Yang, Saghir Hussain, Minlan He, Dequan Gui, Bing Ma, Chaojun Jing, Zhixin Qiao, Changjin Zhu, Qun Yu, 1,2-Benzothiazine 1,1-dioxide carboxylate derivatives as novel potent inhibitors of aldose reductase Bioorganic & Medicinal Chemistry. ,vol. 19, pp. 7262- 7269 ,(2011) , 10.1016/J.BMC.2011.07.051
Katarzyna Gobis, Henryk Foks, Katarzyna Wiśniewska, Maria Dąbrowska-Szponar, Ewa Augustynowicz-Kopeć, Agnieszka Napiórkowska, Synthesis and Antimicrobial Activity of Novel Heterocyclic Sulfamoyl-phenyl-carboximidamides Derived from Clinically Applied Sulfonamides Archiv Der Pharmazie. ,vol. 345, pp. 911- 917 ,(2012) , 10.1002/ARDP.201200160
Günter Kresze, Christoph Seyfried, Achim Trede, Reaktionen mit N‐Sulfinylverbindungen, X1) Benzothiadiazin‐Derivate aus N‐Sulfinyl‐sulfonamiden und N‐Aryl‐amidinen2) European Journal of Organic Chemistry. ,vol. 715, pp. 223- 237 ,(1968) , 10.1002/JLAC.19687150125
Katarzyna Gobis, Henryk Foks, Ewa Augustynowicz-Kopec, Agnieszka Napiorkowska, Malgorzata Szczesio, Andrzej Olczak, Marek L. Glowka, Synthesis, characterization, and tuberculostatic activity of novel 2-(4-nitrobenzoyl)hydrazinecarbodithioic acid derivatives. Monatshefte Fur Chemie. ,vol. 143, pp. 607- 617 ,(2012) , 10.1007/S00706-011-0708-Y