A new facile synthesis of 3-amidoindole derivatives and their evaluation as potential GSK-3β inhibitors
作者： Anahit Pews-Davtyan , Annegret Tillack , Anne-Caroline Schmöle , Stefanie Ortinau , Moritz J. Frech
DOI: 10.1039/B920861E
关键词:
摘要: 3-Amidoindoles were synthesized from commercially available arylhydrazines and propargylamines over Zn-salt mediated one pot procedure in excellent regioselectivity up to 94% yield.
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