TRPM8 ion channel ligands for new therapeutic applications and as probes to study menthol pharmacology
作者： V. Blair Journigan , Nurulain T. Zaveri
DOI: 10.1016/J.LFS.2012.10.032
关键词:
摘要: … have implicated menthol, the natural ligand of TRPM8, in … link between menthol's action via TRPM8 and nicotine … This review gives an overview of reported small-molecule TRPM8 …
sci-hub.se 参考文章(68)
Yi Liu, Ning Qin, TRPM8 in health and disease: cold sensing and beyond. Advances in Experimental Medicine and Biology. ,vol. 704, pp. 185- 208 ,(2011) , 10.1007/978-94-007-0265-3_10
A K Vogt-Eisele, K Weber, M A Sherkheli, G Vielhaber, J Panten, G Gisselmann, H Hatt, Monoterpenoid agonists of TRPV3 British Journal of Pharmacology. ,vol. 151, pp. 530- 540 ,(2007) , 10.1038/SJ.BJP.0707245
Margaret Gardiner-Garden, Daniel E. H. Afar, James G. Kench, Susan M. Henshall, Howard I. Scher, Dorian Willhite, Krishan K. Rasiah, John J. Grygiel, Kurt Gish, David B. Agus, Phillip D. Stricker, Robert L. Sutherland, David I. Quinn, Lisa G. Horvath, David H. Mack, Jordan Hiller, Survival analysis of genome-wide gene expression profiles of prostate cancers identifies new prognostic targets of disease relapse. Cancer Research. ,vol. 63, pp. 4196- 4203 ,(2003)
Mandy Stahre, Kolawole S. Okuyemi, Anne M. Joseph, Steven S. Fu, Racial/ethnic differences in menthol cigarette smoking, population quit ratios and utilization of evidence-based tobacco cessation treatments. Addiction. ,vol. 105, pp. 75- 83 ,(2010) , 10.1111/J.1360-0443.2010.03200.X
David F. Duncan, Sateesh Natarajan, Ofir Moreno, Small-Molecule modulators of TRP-P8 activity ,(2007)
Mark A. Youngman, Raymond W. Colburn, Christopher Flores, Jay Matthews, Laura Reany, Ning Qin, Christopher Teleha, Scott L. Dax, Cold menthol receptor-1 antagonists ,(2007)
Kwokyin Hui, Yibin Guo, Zhong-Ping Feng, Biophysical properties of menthol-activated cold receptor TRPM8 channels. Biochemical and Biophysical Research Communications. ,vol. 333, pp. 374- 382 ,(2005) , 10.1016/J.BBRC.2005.05.123
Giorgio Ortar, Luciano De Petrocellis, Ludovica Morera, Aniello Schiano Moriello, Pierangelo Orlando, Enrico Morera, Marianna Nalli, Vincenzo Di Marzo, (−)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels Bioorganic & Medicinal Chemistry Letters. ,vol. 20, pp. 2729- 2732 ,(2010) , 10.1016/J.BMCL.2010.03.076
Yasuhiro Tsukimi, Kaori Mizuyachi, Tsugiko Yamasaki, Toshiro Niki, Fumihiko Hayashi, Cold response of the bladder in guinea pig: Involvement of transient receptor potential channel, TRPM8 Urology. ,vol. 65, pp. 406- 410 ,(2005) , 10.1016/J.UROLOGY.2004.10.006
Russell L. Stedman, The chemical composition of tobacco and tobacco smoke. Chemical Reviews. ,vol. 68, pp. 153- 207 ,(1968) , 10.1021/CR60252A002