Tandem aza-Wittig reaction/electrocyclic ring-closure a facile entry to the synthesis of fused pyrimidines: preparation of pyrazolo[3,4-d] and 1,2,3-triazolo[4,5-d]pyrimidine derivatives

作者: Pedro Molina , Antonio Arques , Ma Victoria Vinader , Jan Becher , Klaus Brondum

DOI: 10.1016/S0040-4039(00)96536-5

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摘要: Abstract The aza-Wittig reaction of iminophosphoranes derived from 5-azido-4-formyl azoles, with isocyanates or carbon disulfide, leads to functionalized fused pyrimidines.

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