Substrate‐Controlled [5+1] Annulation of 5‐Amino‐1H‐phenylpyrazoles with Alkenes: Divergent Synthesis of Multisubstituted 4,5‐Dihydropyrazolo[1,5‐a]quinazolines

作者: Xunyuan Jiang , Xiaoyi Wei , Fei Lin , Zhixiang Zhang , Guangkai Yao

DOI: 10.1002/EJOC.202000536

关键词:

摘要:

参考文章(30)
Mansi Garg, Monika Chauhan, Pankaj Kumar Singh, Jimi Marin Alex, Raj Kumar, Pyrazoloquinazolines: Synthetic strategies and bioactivities. European Journal of Medicinal Chemistry. ,vol. 97, pp. 444- 461 ,(2015) , 10.1016/J.EJMECH.2014.11.051
Florian Weigend, Reinhart Ahlrichs, Balanced basis sets of split valence, triple zeta valence and quadruple zeta valence quality for H to Rn: Design and assessment of accuracy Physical Chemistry Chemical Physics. ,vol. 7, pp. 3297- 3305 ,(2005) , 10.1039/B508541A
Sabrina Taliani, Isabella Pugliesi, Elisabetta Barresi, Silvia Salerno, Christophe Marchand, Keli Agama, Francesca Simorini, Concettina La Motta, Anna Maria Marini, Francesco Saverio Di Leva, Luciana Marinelli, Sandro Cosconati, Ettore Novellino, Yves Pommier, Roberto Di Santo, Federico Da Settimo, Phenylpyrazolo[1,5-a]quinazolin-5(4H)-one: a suitable scaffold for the development of noncamptothecin topoisomerase I (Top1) inhibitors. Journal of Medicinal Chemistry. ,vol. 56, pp. 7458- 7462 ,(2013) , 10.1021/JM400932C
Chengteh Lee, Weitao Yang, Robert G. Parr, Development of the Colle-Salvetti correlation-energy formula into a functional of the electron density Physical Review B. ,vol. 37, pp. 785- 789 ,(1988) , 10.1103/PHYSREVB.37.785
Kommuri Shekarrao, Partha Pratim Kaishap, Venkateshwarlu Saddanapu, Anthony Addlagatta, Sanjib Gogoi, Romesh C. Boruah, Microwave-assisted palladium mediated efficient synthesis of pyrazolo[3,4-b]pyridines, pyrazolo[3,4-b]quinolines, pyrazolo[1,5-a]pyrimidines and pyrazolo[1,5-a]quinazolines RSC Advances. ,vol. 4, pp. 24001- 24006 ,(2014) , 10.1039/C4RA02865A
Lin Gao, Yunping Song, Xinying Zhang, Shenghai Guo, Xuesen Fan, Copper-catalyzed tandem reactions of 2-bromobenzaldehydes/ketones with aminopyrazoles toward the synthesis of pyrazolo[1,5-a]quinazolines Tetrahedron Letters. ,vol. 55, pp. 4997- 5002 ,(2014) , 10.1016/J.TETLET.2014.07.028
Gabriella Guerrini, Giovanna Ciciani, Samuele Ciattini, Letizia Crocetti, Simona Daniele, Claudia Martini, Fabrizio Melani, Claudia Vergelli, Maria Paola Giovannoni, Pyrazolo[1,5-a]quinazoline scaffold as 5-deaza analogue of pyrazolo[5,1-c][1,2,4]benzotriazine system: synthesis of new derivatives, biological activity on GABAA receptor subtype and molecular dynamic study Journal of Enzyme Inhibition and Medicinal Chemistry. ,vol. 31, pp. 195- 204 ,(2016) , 10.3109/14756366.2015.1014475
Timothy J. Snape, A truce on the Smiles rearrangement: revisiting an old reaction--the Truce-Smiles rearrangement. Chemical Society Reviews. ,vol. 37, pp. 2452- 2458 ,(2008) , 10.1039/B808960D
Stefan Grimme, Jens Antony, Stephan Ehrlich, Helge Krieg, A consistent and accurate ab initio parametrization of density functional dispersion correction (DFT-D) for the 94 elements H-Pu Journal of Chemical Physics. ,vol. 132, pp. 154104- 154104 ,(2010) , 10.1063/1.3382344
Matthew O. Kitching, Timothy E. Hurst, Victor Snieckus, Copper‐Catalyzed Cross‐Coupling Interrupted by an Opportunistic Smiles Rearrangement: An Efficient Domino Approach to Dibenzoxazepinones Angewandte Chemie. ,vol. 51, pp. 2925- 2929 ,(2012) , 10.1002/ANIE.201106786