Synthesis and structure-activity relationship of novel glycylcycline derivatives leading to the discovery of GAR-936

作者: Phaik-Eng Sum , Peter Petersen

DOI: 10.1016/S0960-894X(99)00216-4

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摘要: … synthesis and activity of selected derivatives prepared from minocycline will be discussed, tetracycline and minocycline 1 … These compounds were synthesized via the following synthetic …

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