Compounds and method of identifying, synthesizing, optimizing and profiling protein modulators

摘要: This invention relates to methods of identifying, synthesizing, optimizing and profiling compounds that are inhibitors or activators proteins, both naturally occurring endogenous proteins as well certain variant forms novel identifying such variants. The method accelerates the identification development potential therapeutically effective drugs by simplifying pharmaceutical discovery creation process through improvements in hit identification, lead optimization, biological profiling, rapid elimination toxic compounds. Implementation results overall cost reductions drug resulting from corresponding increases efficiency.