Cycloalkylamines as monoamine reuptake inhibitors
作者： Una Campbell , Liming Shao , John E. Campbell , Sharon Rae Engel , Jianguo Ma
DOI:
关键词: Norepinephrine transporter 、 Medicine 、 Dopamine 、 Monoamine transporter 、 Pharmacology 、 Synaptic cleft 、 Monoamine neurotransmitter 、 Reuptake inhibitor 、 Norepinephrine 、 Reuptake
摘要: The invention relates to novel cyclohexylamine derivatives and their use in the treatment and/or prevention of central nervous system (CNS) disorders, such as depression, anxiety, schizophrenia sleep disorder well methods for synthesis. also pharmaceutical compositions containing compounds invention, inhibiting reuptake endogenous monoamines, dopamine, serotonin norepinephrine from synaptic cleft modulating one or more monoamine transporter.
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