Lysosomal enzyme-cleavable antitumor drug conjugates
作者： Raymond Armand Firestone , Gene Michael Dubowchik
DOI:
关键词: Peptide 、 Drug 、 Ligand (biochemistry) 、 Biochemistry 、 Linker 、 Enzyme 、 A protein 、 Combinatorial chemistry 、 Chemistry 、 Conjugate
摘要: The present invention relates to drug-ligand conjugates wherein the drug is linked ligand through a protein peptide linker and connector, process for preparation of said conjugates, method controlling growth undesirable cells, pharmaceutical compositions, intermediates thereof.
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