Convenient access to substituted acridines by a Buchwald–Hartwig amination
作者： René Csuk , Alexander Barthel , Christian Raschke
DOI: 10.1016/J.TET.2004.05.013
关键词: Chemistry 、 Organic chemistry 、 Buchwald–Hartwig amination 、 Yield (chemistry) 、 Amination 、 Biochemistry 、 Drug discovery
摘要: Abstract A convenient, high yield procedure for the synthesis of anthranilic acids carrying a variety different substituents as well their straightforward transformation into corresponding 9-chloroacridines could be established by using modified Buchwald–Hartwig amination conditions.
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