Quantitative PET Imaging of Tumor Integrin αvβ3 Expression with 18F-FRGD2

作者: Sanjiv S. Gambhir , Weibo Cai , Zhengming Xiong , Xiaoyuan Chen , Yun Wu

DOI:

关键词: In vivoBinding potentialBiochemistryChemistryIntegrin alphaVbeta3Logan plotMolecular imagingIntegrinEx vivoBiophysicsReceptor

摘要: … new therapeutic drugs with favorable tumor targeting and in vivo kinetics. … c(RGDyK)] 2 with 18 F and evaluated its tumor-targeting efficacy and pharmacokinetics of 18 F-FB–E[c(RGDyK…

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