Solvent-free synthesis of azole carboximidamides

作者: Sotir Zahariev , Corrado Guarnaccia , Doriano Lamba , Maša Čemažar , Sándor Pongor

DOI: 10.1016/J.TETLET.2004.10.114

关键词:

摘要: A one-pot procedure is described for the preparation of 1H-pyrazole-carboximidamides 2, 1 H-benzotriazole-carboximidamides 3 and guanidinylation amines with 3. The X-ray crystal structure N,N-dimethyl- H-benzotriazole- -carboximidamide 3b, has been determined. (C) 2004 Elsevier Ltd. All rights reserved.

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