Generic GPCR residue numbers – aligning topology maps while minding the gaps
作者： Vignir Isberg , Chris de Graaf , Andrea Bortolato , Vadim Cherezov , Vsevolod Katritch
DOI: 10.1016/J.TIPS.2014.11.001
关键词:
摘要: Generic residue numbers facilitate comparisons of, for example, mutational effects, ligand interactions, and structural motifs. The numbering scheme by Ballesteros and Weinstein for …
ru.nl
narcis.nl
elsevier.com
core.ac.uk 参考文章(77)
Tsviya Olender, Noam Nativ, Doron Lancet, HORDE: Comprehensive Resource for Olfactory Receptor Genomics Methods of Molecular Biology. ,vol. 1003, pp. 23- 38 ,(2013) , 10.1007/978-1-62703-377-0_2
Yoshikazu Katao, Takahiro Seki, Masamichi Satoh, Yasuhide Aoki, Tatsuhiro Onogi, Masabumi Minami, Seishi Katsumata, Takayuki Nakagawa, A single residue, Lys108, of the delta-opioid receptor prevents the mu-opioid-selective ligand [D-Ala2,N-MePhe4,Gly-ol5]enkephalin from binding to the delta-opioid receptor. Molecular Pharmacology. ,vol. 50, pp. 1413- 1422 ,(1996)
Kolakowski Lf, GCRDB: A G-PROTEIN-COUPLED RECEPTOR DATABASE Receptors & Channels. ,vol. 2, pp. 1- 7 ,(1994)
J.M. Baldwin, The probable arrangement of the helices in G protein‐coupled receptors. The EMBO Journal. ,vol. 12, pp. 1693- 1703 ,(1993) , 10.1002/J.1460-2075.1993.TB05814.X
Andrea Bortolato, Andrew S Doré, Kaspar Hollenstein, Benjamin G Tehan, Jonathan S Mason, Fiona H Marshall, Structure of Class B GPCRs: new horizons for drug discovery British Journal of Pharmacology. ,vol. 171, pp. 3132- 3145 ,(2014) , 10.1111/BPH.12689
A J Kooistra, S Kuhne, I J P de Esch, R Leurs, C de Graaf, A structural chemogenomics analysis of aminergic GPCRs: lessons for histamine receptor ligand design British Journal of Pharmacology. ,vol. 170, pp. 101- 126 ,(2013) , 10.1111/BPH.12248
Kristen L. Pierce, Richard T. Premont, Robert J. Lefkowitz, Seven-transmembrane receptors. Nature Reviews Molecular Cell Biology. ,vol. 3, pp. 639- 650 ,(2002) , 10.1038/NRM908
DJ Scholten, M Canals, D Maussang, L Roumen, MJ Smit, M Wijtmans, C de Graaf, HF Vischer, R Leurs, Pharmacological modulation of chemokine receptor function British Journal of Pharmacology. ,vol. 165, pp. 1617- 1643 ,(2012) , 10.1111/J.1476-5381.2011.01551.X
Juan A. Ballesteros, Harel Weinstein, [19] Integrated methods for the construction of three-dimensional models and computational probing of structure-function relations in G protein-coupled receptors Methods in Neurosciences. ,vol. 25, pp. 366- 428 ,(1995) , 10.1016/S1043-9471(05)80049-7
John P. Overington, Bissan Al-Lazikani, Andrew L. Hopkins, How many drug targets are there Nature Reviews Drug Discovery. ,vol. 5, pp. 993- 996 ,(2006) , 10.1038/NRD2199