Inhibitory activities of indolizine derivatives: a patent review.

作者: Kamal M. Dawood , Ashraf A. Abbas

DOI: 10.1080/13543776.2020.1798402

关键词:

摘要: Indolizines are structural isomers with indoles. Although several indole-based commercial drugs available in the market, none of indolizine-based up-to-date. Natural and...

参考文章(120)
Liliana Lucescu, Alina Ghinet, Dalila Belei, Benoît Rigo, Joëlle Dubois, Elena Bîcu, Discovery of indolizines containing triazine moiety as new leads for the development of antitumoral agents targeting mitotic events Bioorganic & Medicinal Chemistry Letters. ,vol. 25, pp. 3975- 3979 ,(2015) , 10.1016/J.BMCL.2015.07.025
Kevin Hodgetts, Jun Yuan, Qin Guo, David C. Ihle, Heteroaryl amide analogues as p2x7 antagonists ,(2008)
Duncan A. Hay, Catherine M. Rogers, Oleg Fedorov, Cynthia Tallant, Sarah Martin, Octovia P. Monteiro, Susanne Müller, Stefan Knapp, Christopher J. Schofield, Paul E. Brennan, Design and synthesis of potent and selective inhibitors of BRD7 and BRD9 bromodomains MedChemComm. ,vol. 6, pp. 1381- 1386 ,(2015) , 10.1039/C5MD00152H
Won-Gil Lee, Kathleen M. Frey, Ricardo Gallardo-Macias, Krasimir A. Spasov, Albert H. Chan, Karen S. Anderson, William L. Jorgensen, Discovery and crystallography of bicyclic arylaminoazines as potent inhibitors of HIV-1 reverse transcriptase. Bioorganic & Medicinal Chemistry Letters. ,vol. 25, pp. 4824- 4827 ,(2015) , 10.1016/J.BMCL.2015.06.074
M. Iqbal Choudhary, Sarfraz Ahmad Nawaz, Zaheer-ul-Haq, M. Kamran Azim, M. Nabeel Ghayur, M. Arif Lodhi, Saima Jalil, Asaad Khalid, Amir Ahmed, Bernd M. Rode, Atta-ur-Rahman, Anwar-ul-Hassan Gilani, Viqar Uddin Ahmad, Juliflorine: a potent natural peripheral anionic-site-binding inhibitor of acetylcholinesterase with calcium-channel blocking potential, a leading candidate for Alzheimer's disease therapy. Biochemical and Biophysical Research Communications. ,vol. 332, pp. 1171- 1179 ,(2005) , 10.1016/J.BBRC.2005.05.068
Abhijit Hazra, Shyamal Mondal, Arindam Maity, Subhendu Naskar, Pritam Saha, Rupankar Paira, Krishnendu B Sahu, Priyankar Paira, Soma Ghosh, Chandrima Sinha, Amalesh Samanta, Sukdeb Banerjee, Nirup B Mondal, None, Amberlite-IRA-402 (OH) ion exchange resin mediated synthesis of indolizines, pyrrolo [1,2-a] quinolines and isoquinolines: antibacterial and antifungal evaluation of the products. European Journal of Medicinal Chemistry. ,vol. 46, pp. 2132- 2140 ,(2011) , 10.1016/J.EJMECH.2011.02.066
Wenlin Huang, Tao Zuo, Xiao Luo, Hongwei Jin, Zhenming Liu, Zhenjun Yang, Xianghui Yu, Liangren Zhang, Lihe Zhang, Indolizine derivatives as HIV-1 VIF-ElonginC interaction inhibitors. Chemical Biology & Drug Design. ,vol. 81, pp. 730- 741 ,(2013) , 10.1111/CBDD.12119
Sandrine Gerber-Lemaire, Lucienne Juillerat-Jeanneret, Studies toward new anti-cancer strategies based on alpha-mannosidase inhibition. Chimia. ,vol. 64, pp. 634- 639 ,(2010) , 10.2533/CHIMIA.2010.634
Nam Doo Kim, Eun-Sook Park, Young Hoon Kim, Seung Kee Moon, Sung Sook Lee, Soon Kil Ahn, Dae-Yeul Yu, Kyoung Tai No, Kyun-Hwan Kim, Structure-based virtual screening of novel tubulin inhibitors and their characterization as anti-mitotic agents Bioorganic & Medicinal Chemistry. ,vol. 18, pp. 7092- 7100 ,(2010) , 10.1016/J.BMC.2010.07.072