Mutant-Selective Allosteric EGFR Degraders are Effective Against a Broad Range of Drug-Resistant Mutations.

作者: Jaebong Jang , Ciric To , Dries J. H. De Clercq , Eunyoung Park , Charles M. Ponthier

DOI: 10.1002/ANIE.202003500

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摘要: … or DDC-01-163 alone or in combination with two constant doses of DDC-01-163 and … Our results showed that the addition of both 0.01 μm and 0.1 μm of DDC-01-163 shifted the …

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