Method for determining drug compositions to prevent desensitization of cellular receptors

摘要: Drug compositions combining antagonists with agonists to prevent desensitization of cellular receptors. An agonist is a substance or drug that produces maximal nearly response, whereas an antagonist molecule no but can block the action agonist/drug. A partial moderate response and also receptor The instant invention solves problem determining optimal concentration inhibitor which necessary desensitization, without causing unnecessary unwanted inhibition, by providing formulative method detailing how competitive should be combined in specific proportion maximize maintain throughout therapy/administration.