Neratinib for the treatment of HER2-positive early stage breast cancer.

作者: Isabel Echavarria , Sara López-Tarruella , Iván Márquez-Rodas , Yolanda Jerez , Miguel Martin

DOI: 10.1080/14737140.2017.1338954

关键词:

摘要: … Neratinib activity relies on its covalent binding and blockade … Neratinib forms a covalent bond with this cysteine residue, … or serine–threonine kinases, such as c-met, src, or Kdr. Neratinib …

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