Palladium‐Catalyzed Direct Arylations of 1,2,3‐Triazoles with Aryl Chlorides using Conventional Heating
作者： Lutz Ackermann , Rubén Vicente , Robert Born
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摘要: Generally applicable, palladium-catalyzed direct arylations of 1,2,3-triazoles with aryl chlorides were accomplished through conventional heating at reaction temperatures 105-120 °C. Thereby, intra-and intermolecular C-H bond functionalizations achieved a variety differently substituted as electrophiles, bearing numerous valuable functional groups.
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